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Metoprolol

Lopressor, Toprol-XL

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Meta Information

ID:metoprolol
Name:Metoprolol
Schema Version:1.5

Alternate Names

  • Lopressor
  • Toprol-XL

Active Compound

metoprolol

Intervention Type

therapeutic_agent

Delivery

Route:
oral
Scope:
  • systemic

Regulatory Status

  • us:rx_drug
  • eu:rx_drug

Indication

Focus:
disease_treatment
Description:
Treatment of hypertension (high blood pressure), angina (chest pain), and heart failure to improve survival after a heart attack.

Typical Protocol

  • For hypertension, typically started at 25-100 mg daily in one or two divided doses.
  • For stable angina, the usual initial dosage is 100 mg daily in two divided doses.
  • For heart failure, dosing is started very low (e.g., 12.5 mg daily) and titrated up slowly under supervision.

Expected Cost Mean

Low Cost:
5
High Cost:
30
Cost Type:
monthly
Description:
Generic prescription cost, which is typically covered by insurance.

Summary

Metoprolol is a selective beta-1 adrenergic receptor blocker, or 'beta-blocker'. It works primarily by decreasing the heart's workload, which lowers heart rate, reduces the force of heart contractions, and lowers blood pressure. Its role is strictly for the management of diagnosed cardiovascular diseases, not for general healthspan extension in healthy individuals.

Purpose

Manages cardiovascular disease by reducing heart rate and blood pressure.

Card Summary

A beta-blocker medication used to treat high blood pressure, chest pain (angina), and heart failure by reducing cardiac workload.

Drug Class

beta_blockers

Drugs In Class

Empty Array

Impact

Score:
8.5
Justification:
Foundational, first-line therapy for managing hypertension, angina, and post-heart attack care.

Evidence

Grade:
A
Score:
10
Justification:
Extensive, multi-decade evidence from numerous large-scale human RCTs and meta-analyses.

Safety

Score:
5.5
Justification:
Well-established side effect profile; requires medical supervision for dose titration and monitoring.

Flags

  • Abrupt discontinuation can cause rebound hypertension or cardiac events.
  • May mask symptoms of hypoglycemia in diabetic patients.
  • Can worsen symptoms of asthma or COPD.
  • Common side effects include fatigue, dizziness, depression, and bradycardia (slow heart rate).
  • Contraindicated in patients with severe bradycardia, heart block, or cardiogenic shock.

Verdict

Highly effective for cardiovascular disease management under medical supervision.

Qualifier

scope: systemic, focused on disease treatment

Created

2026-05-02T01:57:50.814315Z

Ai Model

Gemini 2.5 Pro (High)

Non Healthspan

True